Synthesis of Diiodo-Functionalized Benzo[b]furans via Electrophilic Iodocyclization

AUTOR(ES)

Frota, Carlise, Rossini, Allan F. C., Casagrande, Gleison A., Pizzuti, Lucas, Raminelli, Cristiano

FONTE

J. Braz. Chem. Soc.

DATA DE PUBLICAÇÃO

2017-10

RESUMO

An electrophilic iodocyclization reaction involving alkynylated 2-iodoanisoles and molecular iodine in the presence of sodium bicarbonate was developed and diiodo-functionalized benzo[b]furans were obtained in yields from 45 to 99%.

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